ReN-1869 hydrochloride Catalog No.:M19898-C Smiles: CSCCC(NC(=O)C(N)CS)C(=O)N1CCCC1C(=O)NC(CC(C)C)C(=O)NC(CC1=CN=CN1)C(=O)NC(CO)C(=O)NC(CCCN=C(N)N)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)NC(CC1C=CC=CC=1)C(=O)N1CCCC1C(O)=O

Smiles: CSCCC(NC(=O)C(N)CS)C(=O)N1CCCC1C(=O)NC(CC(C)C)C(=O)NC(CC1=CN=CN1)C(=O)NC(CO)C(=O)NC(CCCN=C(N)N)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)NC(CC1C=CC=CC=1)C(=O)N1CCCC1C(O)=O

a transcriptional repressor target at transcription factor E2F-1

Functional assays

Chemical Name: 2-amino-3-methyl-N-[2-(morpholin-4-yl)ethyl]pentanamide

with 50% effective concentrations ranging between 4 and 71 nM

ReN-1869 hydrochloride Catalog No.:M19898-C Smiles: CSCCC(NC(=O)C(N)CS)C(=O)N1CCCC1C(=O)NC(CC(C)C)C(=O)NC(CC1=CN=CN1)C(=O)NC(CO)C(=O)NC(CCCN=C(N)N)C(=O)NC(C(C)C)C(=O)N1CCCC1C(=O)NC(CC1C=CC=CC=1)C(=O)N1CCCC1C(O)=OReN 1869 hydrochloride is a novel, selective histamine H1 receptor antagonist, which demonstrates affinity to the histamine H1 receptor (guinea pig brain) with Ki of 0. 190. 04 M and the non selective site (guinea pig brain) with Ki of 0. 45 M. Product information CAS Number: 170149 76 5 Molecular Weight: 397. 94 Formula: C24H28ClNO2 Chemical Name: (3R) 1 (3 {tricyclo[9. 4. 0. 0,]pentadeca 1(15),3,5,7,11,13 hexaen 2 ylidene}propyl)piperidine 3